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Minaprine
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Clinical data | |
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AHFS/Drugs.com | International Drug Names |
Routes of administration |
Oral |
ATC code | |
Legal status | |
Legal status |
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Pharmacokinetic data | |
Elimination half-life | 2-2.5 hours |
Identifiers | |
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CAS Number | |
PubChem CID | |
ChemSpider |
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ChEMBL | |
CompTox Dashboard (EPA) | |
ECHA InfoCard | 100.043.012 |
Chemical and physical data | |
Formula | C17H22N4O |
Molar mass | 298.390 g·mol−1 |
3D model (JSmol) | |
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NY (what is this?) (verify) |
Minaprine (INN, USAN, BAN) (brand names Brantur, Cantor) is a monoamine oxidase inhibitor antidepressant drug that was used in France for the treatment of depression until it was withdrawn from the market in 1996 because it caused convulsions.
A study found that it acts as a reversible inhibitor of MAO-A (RIMA) in rats. In a study it has also been found to weakly inhibit acetylcholinesterase in rat brain (striatum) homogenates.
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Phenethylamines (dopamine, epinephrine, norepinephrine) |
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