Eprobemide
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| Clinical data | |
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| Trade names | Befol (RU) |
| Other names | Befol |
| Routes of administration |
Oral |
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| Chemical and physical data | |
| Formula | C14H19ClN2O2 |
| Molar mass | 282.77 g·mol−1 |
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Eprobemide (INN) is a pharmaceutical drug that was used as an antidepressant in Russia (under the brand name Бефол/Befol). It is a non-competitive reversible inhibitor of monoamine oxidase A that exhibits selective action on serotonin deamination. Eprobemide differs from moclobemide only in the linker that connects the morpholine fragment with the chlorobenzamide — moclobemide has two carbon atoms while eprobemide has three. Its registration was cancelled on December 30, 2003.
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| Non-specific |
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Phenethylamines (dopamine, epinephrine, norepinephrine) |
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Tryptamines (serotonin, melatonin) |
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| Histamine |
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