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Abandoned drugs
Bexlosteride
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    Bexlosteride

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    Bexlosteride
    Bexlosteride.svg
    Clinical data
    Other names LY 300502
    Routes of
    administration    		 Oral
    ATC code
    • none
    Legal status
    Legal status
    • In general: uncontrolled
    Identifiers
    • (4aR,10bR)-8-Chloro-4-methyl-1,4,4a,5,6,10b-hexahydrobenzo[f]quinolin-3(2H)-one
    CAS Number
    PubChem CID
    ChemSpider
    UNII
    ChEMBL
    Chemical and physical data
    Formula C14H16ClNO
    Molar mass 249.74 g·mol−1
    3D model (JSmol)
    • CN1[C@@H]2CCc3cc(ccc3[C@H]2CCC1=O)Cl
    • InChI=1S/C14H16ClNO/c1-16-13-6-2-9-8-10(15)3-4-11(9)12(13)5-7-14(16)17/h3-4,8,12-13H,2,5-7H2,1H3/t12-,13-/m1/s1 checkY
    • Key:WQBIOEFDDDEARX-CHWSQXEVSA-N checkY
     ☒NcheckY (what is this?)  (verify)

    Bexlosteride is a potent and noncompetitive inhibitor of the enzyme 5α-reductase related to finasteride and dutasteride. It is selective for the type I isoform of the enzyme. It advanced to Phase III clinical trials, but development was halted at that stage, and it was never marketed.

    See also


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