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Abandoned drugs
Bolmantalate
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    Bolmantalate

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    Bolmantalate
    Bolmantalate.svg
    Clinical data
    Other names LY-38851; Lilly 38851; Nandrolone adamantoate; Nandrolone adamantane-1-carboxylate; 19-Nortestosterone 17β-adamantoate
    Routes of
    administration    		 Intramuscular injection
    Drug class Androgen; Anabolic steroid; Androgen ester; Progestogen
    Identifiers
    • [(8R,9S,10R,13S,14S,17S)-13-methyl-3-oxo-2,6,7,8,9,10,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl] adamantane-1-carboxylate
    CAS Number
    PubChem CID
    ChemSpider
    UNII
    KEGG
    ChEMBL
    CompTox Dashboard (EPA)
    Chemical and physical data
    Formula C29H40O3
    Molar mass 436.636 g·mol−1
    3D model (JSmol)
    • C[C@]12CC[C@H]3[C@H]([C@@H]1CC[C@@H]2OC(=O)C45CC6CC(C4)CC(C6)C5)CCC7=CC(=O)CC[C@H]37
    • InChI=1S/C29H40O3/c1-28-9-8-23-22-5-3-21(30)13-20(22)2-4-24(23)25(28)6-7-26(28)32-27(31)29-14-17-10-18(15-29)12-19(11-17)16-29/h13,17-19,22-26H,2-12,14-16H2,1H3/t17?,18?,19?,22-,23+,24+,25-,26-,28-,29?/m0/s1
    • Key:NCXAMLZZPQRJGY-PVAKYVEVSA-N

    Bolmantalate (developmental code name LY-38851 or Lilly 38851), also known as 19-nortestosterone 17β-adamantoate (or nandrolone adamantoate), is an androgen and anabolic steroid and a nandrolone ester which was synthesized and developed by Eli Lilly in 1865 but was never marketed.

    Relative affinities (%) of nandrolone and related steroids
    Compound PR AR ER GR MR SHBG CBG
    Nandrolone 20 154–155 <0.1 0.5 1.6 1–16 0.1
    Testosterone 1.0–1.2 100 <0.1 0.17 0.9 19–82 3–8
    Estradiol 2.6 7.9 100 0.6 0.13 8.7–12 <0.1
    Notes: Values are percentages (%). Reference ligands (100%) were progesterone for the PR, testosterone for the AR, estradiol for the ER, dexamethasone for the GR, aldosterone for the MR, dihydrotestosterone for SHBG, and cortisol for CBG. Sources: See template.

    See also




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