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Mu-opioid receptor agonists
LS-115509
Другие языки:

    LS-115509

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    LS-115509
    LS-115509 Structure.svg
    Clinical data
    ATC code
    • none
    Identifiers
    • 4-ethoxy-4-(furan-2-yl)-3-methyl-1-(2-phenylethyl)piperidine
    CAS Number
    PubChem CID
    ChemSpider
    UNII
    CompTox Dashboard (EPA)
    Chemical and physical data
    Formula C20H27NO2
    Molar mass 313.441 g·mol−1
    3D model (JSmol)
    • CCOC1(CCN(CC1C)CCC2=CC=CC=C2)C3=CC=CO3
    • InChI=1S/C20H27NO2/c1-3-23-20(19-10-7-15-22-19)12-14-21(16-17(20)2)13-11-18-8-5-4-6-9-18/h4-10,15,17H,3,11-14,16H2,1-2H3
    • Key:INLMDDDTZIKNNI-UHFFFAOYSA-N

    LS-115509 is an opioid analgesic related to the 4-phenylpiperidine family. It is comparable to drugs such as prodine and pheneridine, but is distinguished by the presence of an ether group and furan ring at the piperidine 4-position, which are not found in other drugs of this class. In animal studies, it has around 2-3x the potency of morphine depending on what assay is used. Like prodine, it has two stereocenters and four possible enantiomers, but the activity of these has not been tested separately.

    See also




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